Carbutamide

Chemical compound
  • A10BB06 (WHO)
Identifiers
  • 4-amino-N-(butylcarbamoyl)benzenesulfonamide
CAS Number
  • 339-43-5 checkY
PubChem CID
  • 9564
ChemSpider
  • 9189 ☒N
UNII
  • E3K8P4869P
ChEMBL
  • ChEMBL448570 checkY
CompTox Dashboard (EPA)
  • DTXSID8022741 Edit this at Wikidata
ECHA InfoCard100.005.841 Edit this at WikidataChemical and physical dataFormulaC11H17N3O3SMolar mass271.33 g·mol−13D model (JSmol)
  • Interactive image
  • O=S(=O)(c1ccc(N)cc1)NC(=O)NCCCC
InChI
  • InChI=1S/C11H17N3O3S/c1-2-3-8-13-11(15)14-18(16,17)10-6-4-9(12)5-7-10/h4-7H,2-3,8,12H2,1H3,(H2,13,14,15) ☒N
  • Key:VDTNNGKXZGSZIP-UHFFFAOYSA-N ☒N
 ☒NcheckY (what is this?)  (verify)

Carbutamide (brand name Glucidoral) is an anti-diabetic drug of the sulfonylurea class, developed by Servier.

It is classified as first-generation.[1]

It was patented in 1953 and approved for medical use in 1956.[2]

See also

  • Hellmuth Kleinsorge (1920-2001) German medical doctor

References

  1. ^ Ballagi-Pordány G, Köszeghy A, Koltai MZ, Aranyi Z, Pogátsa G (January 1990). "Divergent cardiac effects of the first and second generation hypoglycemic sulfonylurea compounds". Diabetes Research and Clinical Practice. 8 (2): 109–114. doi:10.1016/0168-8227(90)90020-T. PMID 2106423.
  2. ^ Fischer J, Ganellin CR (2006). Analogue-based Drug Discovery. John Wiley & Sons. p. 449. ISBN 9783527607495.
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